Description
malaria
blood-schizontocidals
falcipain inhibition
hemozoin biomineralization
Main Local Researcher
Coordination
Faculdade de Ciências da Universidade do Porto (FCUP/UP)
Partners
Universidade de Aveiro (UA)
link
http://www.fct.pt/apoios/projectos/consulta/vglobal_projecto?idProjecto=116864&idElemConcurso=4144
Outputs
N-Cinnamoylation of Antimalarial Classics: Quinacrine Analogues with Decreased Toxicity and Dual-Stage Activity
Gomes, A; Perez, B; Albuquerque, I; Machado, M; Prudencio, M; Nogueira, F; Teixeira, C; Gomes, PIn vitro efficiency of 9-(N-cinnamoylbutyl)aminoacridines against blood- and liver-stage malaria parasites
Perez, B; Teixeira, C; Gomes, AS; Albuquerque, IS; Gut, J; Rosenthal, PJ; Prudencio, M; Gomes, PRecycling antimalarial leads for cancer: Antiproliferative properties of N-cinnamoyl chloroquine analogues
Perez, BC; Fernandes, I; Mateus, N; Teixeira, C; Gomes, PN-Cinnamoylated Chloroquine Analogues as Dual-Stage Antimalarial Leads
Perez, BC; Teixeira, C; Albuquerque, IS; Gut, J; Rosenthal, PJ; Gomes, JRB; Prudencio, M; Gomes, PPRIMACINS, N-cinnamoyl-primaquine conjugates, with improved liver-stage antimalarial activity
Perez, B; Teixeira, C; Albuquerque, IS; Gut, J; Rosenthal, PJ; Prudencio, M; Gomes, PCinnamic Acid/Chloroquinoline Conjugates as Potent Agents against Chloroquine-Resistant Plasmodium falciparum
Perez, B; Teixeira, C; Gut, J; Rosenthal, PJ; Gomes, JRB; Gomes, PNovel cinnamic acid/4-aminoquinoline conjugates bearing non-proteinogenic amino acids: Towards the development of potential dual action antimalarials
Perez, BC; Teixeira, C; Figueiras, M; Gut, J; Rosenthal, PJ; Gomes, JRB; Gomes, PSponsors
